Kamil Musilek : rechercher sur Z-Library

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1

In Vitro Ability of Currently Available Oximes to Reactivate Organophosphate Pesticide-Inhibited Human Acetylcholinesterase and Butyrylcholinesterase

Jun, Daniel, Musilova, Lucie, Musilek, Kamil, Kuca, Kamil

Journal:

International Journal of Molecular Sciences

Année:

2011

Langue:

english

Fichier:

PDF, 185 KB

english, 2011

2

ChemInform Abstract: Design, Evaluation and Structure—Activity Relationship Studies of the AChE Reactivators Against Organophosphorus Pesticides

Kamil Musilek, Martin Dolezal, Frank Gunn-Moore, Kamil Kuca

Journal:

Année:

2011

Fichier:

PDF, 18 KB

2011

3

Monooxime-monocarbamoyl Bispyridinium Xylene-Linked Reactivators of Acetylcholinesterase—Synthesis, In vitro and Toxicity Evaluation, and Docking Studies

Kamil Musilek, Ondrej Holas, Jan Misik, Miroslav Pohanka, Ladislav Novotny, Vlastimil Dohnal, Veronika Opletalova, Kamil Kuca

Journal:

Année:

2010

Langue:

english

Fichier:

PDF, 525 KB

english, 2010

4

Synthesis of monooxime-monocarbamoyl bispyridinium compounds bearing ( E )-but-2-ene linker and evaluation of their reactivation activity against tabun- and paraoxon-inhibited acetylcholinesterase

Musilek, Kamil, Holas, Ondrej, Kuca, Kamil, Jun, Daniel, Dohnal, Vlastimil, Opletalova, Veronika, Dolezal, Martin

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Année:

2008

Langue:

english

Fichier:

PDF, 179 KB

english, 2008

5

In vitro identification of novel acetylcholinesterase reactivators

Kuca, Kamil, RC, Gupta, Musilek, Kamil, Jun, Daniel, Pohanka, Miroslav

Journal:

Année:

2009

Langue:

english

Fichier:

PDF, 763 KB

english, 2009

6

Redox- and non-redox-metal-induced formation of free radicals and their role in human disease

Valko, Marian, Jomova, Klaudia, Rhodes, Christopher J., Kuča, Kamil, Musílek, Kamil

Journal:

Archives of Toxicology

Année:

2016

Langue:

english

Fichier:

PDF, 1.66 MB

english, 2016

7

Design, synthesis and in vitro evaluation of benzothiazole-based ureas as potential ABAD/17β-HSD10 modulators for Alzheimer’s disease treatment

Hroch, Lukas, Benek, Ondrej, Guest, Patrick, Aitken, Laura, Soukup, Ondrej, Janockova, Jana, Musil, Karel, Dohnal, Vlastimil, Dolezal, Rafael, Kuca, Kamil, Smith, Terry K, Gunn-Moore, Frank, Musilek,

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2016

Langue:

english

Fichier:

PDF, 347 KB

english, 2016

8

Vector Control and Insecticidal Resistance in the African Malaria Mosquito Anopheles gambiae

Schmidt, Monika, Hrabcova, Veronika, Jun, Daniel, Kuca, Kamil, Musilek, Kamil

Journal:

Chemical Research in Toxicology

Année:

2018

Langue:

english

Fichier:

PDF, 1.48 MB

english, 2018

9

Taking advantage of cellular uptake of ferritin nanocages for targeted drug delivery

Tesarova, Barbora, Musilek, Kamil, Rex, Simona, Heger, Zbynek

Journal:

Journal of Controlled Release

Année:

2020

Fichier:

PDF, 9.07 MB

2020

10

ChemInform Abstract: Synthesis and in vitro Evaluation of New Tacrine Derivatives-bis-alkylene Linked 7-MEOTA.

Jan Korabecny, Ondrej Holas, Kamil Musilek, Miroslav Pohanka, Veronika Opletalova, Vlastimil Dohnal, Kamil Kuca

Journal:

Année:

2010

Fichier:

PDF, 22 KB

2010

11

Effective bisquaternary reactivators of tabun-inhibited AChE

Kamil Kuca, Jiri Cabal, Kamil Musilek, Daniel Jun, Jiri Bajgar

Journal:

Journal of Applied Toxicology

Année:

2005

Langue:

english

Fichier:

PDF, 126 KB

english, 2005

12

Effect of five acetylcholinesterase reactivators on tabun-intoxicated rats: induction of oxidative stress versus reactivation efficacy

Miroslav Pohanka, Jana Zdarova Karasova, Kamil Musilek, Kamil Kuca, Jiri Kassa

Journal:

Journal of Applied Toxicology

Année:

2009

Langue:

english

Fichier:

PDF, 337 KB

english, 2009

13

Design, evaluation and structure—Activity relationship studies of the AChE reactivators against organophosphorus pesticides

Kamil Musilek, Martin Dolezal, Frank Gunn-Moore, Kamil Kuca

Journal:

Medicinal Research Reviews

Année:

2011

Langue:

english

Fichier:

PDF, 372 KB

english, 2011

14

Corrigendum: Design, evaluation and structure—activity relationship studies of the AChE reactivators against organophosphorus pesticides

Kamil Musilek, Martin Dolezal, Frank Gunn-Moore, Kamil Kuca

Journal:

Medicinal Research Reviews

Année:

2011

Langue:

english

Fichier:

PDF, 51 KB

english, 2011

15

Novel series of bispyridinium compounds bearing a (Z)-but-2-ene linker—Synthesis and evaluation of their reactivation activity against tabun and paraoxon-inhibited acetylcholinesterase

Kamil Musilek, Ondrej Holas, Kamil Kuca, Daniel Jun, Vlastimil Dohnal, Veronika Opletalova, Martin Dolezal

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2007

Langue:

english

Fichier:

PDF, 216 KB

english, 2007

16

Monooxime reactivators of acetylcholinesterase with (E)-but-2-ene linker—Preparation and reactivation of tabun- and paraoxon-inhibited acetylcholinesterase

Kamil Musilek, Ondrej Holas, Daniel Jun, Vlastimil Dohnal, Frank Gunn-Moore, Veronika Opletalova, Martin Dolezal, Kamil Kuca

Journal:

Bioorganic & Medicinal Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 207 KB

english, 2007

17

Monoquaternary pyridinium salts with modified side chain—synthesis and evaluation on model of tabun- and paraoxon-inhibited acetylcholinesterase

Kamil Musilek, Jiri Kucera, Daniel Jun, Vlastimil Dohnal, Veronika Opletalova, Kamil Kuca

Journal:

Bioorganic & Medicinal Chemistry

Année:

2008

Langue:

english

Fichier:

PDF, 202 KB

english, 2008

18

Fluorinated pyridinium oximes as potential reactivators for acetylcholinesterases inhibited by paraoxon organophosphorus agent

Hee Chun Jeong, No-Joong Park, Chong Hak Chae, Kamil Musilek, Jiri Kassa, Kamil Kuca, Young-Sik Jung

Journal:

Bioorganic & Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 259 KB

english, 2009

19

Mono-oxime bisquaternary acetylcholinesterase reactivators with prop-1,3-diyl linkage—Preparation, in vitro screening and molecular docking

Kamil Musilek, Marketa Komloova, Ondrej Holas, Anna Horova, Miroslav Pohanka, Frank Gunn-Moore, Vlastimil Dohnal, Martin Dolezal, Kamil Kuca

Journal:

Bioorganic & Medicinal Chemistry

Année:

2011

Langue:

english

Fichier:

PDF, 505 KB

english, 2011

20

Preparation and in vitro screening of symmetrical bispyridinium cholinesterase inhibitors bearing different connecting linkage—initial study for Myasthenia gravis implications

Kamil Musilek, Marketa Komloova, Vlasta Zavadova, Ondrej Holas, Martina Hrabinova, Miroslav Pohanka, Vlastimil Dohnal, Florian Nachon, Martin Dolezal, Kamil Kuca, Young-Sik Jung

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 279 KB

english, 2010

21

Synthesis and in vitro evaluation of N-alkyl-7-methoxytacrine hydrochlorides as potential cholinesterase inhibitors in Alzheimer disease

Jan Korabecny, Kamil Musilek, Ondrej Holas, Jiri Binder, Filip Zemek, Jan Marek, Miroslav Pohanka, Veronika Opletalova, Vlastimil Dohnal, Kamil Kuca

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 580 KB

english, 2010

22

Preparation, in vitro screening and molecular modelling of symmetrical 4-tert-butylpyridinium cholinesterase inhibitors—Analogues of SAD-128

Kamil Musilek, Jan Roder, Marketa Komloova, Ondrej Holas, Martina Hrabinova, Miroslav Pohanka, Vlastimil Dohnal, Veronika Opletalova, Kamil Kuca, Young-Sik Jung

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 562 KB

english, 2011

23

Preparation, in vitro screening and molecular modelling of symmetrical bis-quinolinium cholinesterase inhibitors—implications for early Myasthenia gravis treatment

Marketa Komloova, Kamil Musilek, Anna Horova, Ondrej Holas, Vlastimil Dohnal, Frank Gunn-Moore, Kamil Kuca

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 542 KB

english, 2011

24

Preparation and in vitro screening of symmetrical bis-isoquinolinium cholinesterase inhibitors bearing various connecting linkage – Implications for early Myasthenia gravis treatment

Kamil Musilek, Marketa Komloova, Ondrej Holas, Martina Hrabinova, Miroslav Pohanka, Vlastimil Dohnal, Florian Nachon, Martin Dolezal, Kamil Kuca

Journal:

European Journal of Medicinal Chemistry

Année:

2011

Langue:

english

Fichier:

PDF, 512 KB

english, 2011

25

An evaluation of therapeutic and reactivating effects of newly developed oximes (K156, K203) and commonly used oximes (obidoxime, trimedoxime, HI-6) in tabun-poisoned rats and mice

Jiri Kassa, Jana Karasova, Kamil Musilek, Kamil Kuca

Journal:

Année:

2008

Langue:

english

Fichier:

PDF, 184 KB

english, 2008

26

Penetration of polar organic compounds through the blood-brain barrier

Huba Kalász, Kamil Musílek, Kornélia Tekes

Journal:

BMC Pharmacology

Année:

2011

Langue:

english

Fichier:

PDF, 75 KB

english, 2011

27

In vitroreactivation potency of acetylcholinesterase reactivators — K074 and K075 — to reactivate tabun-inhibited human brain cholinesterases

Kamil Kuca, Jiri Cabal, Daniel Jun, Kamil Musilek

Journal:

Neurotoxicity Research

Année:

2007

Langue:

english

Fichier:

PDF, 873 KB

english, 2007

28

RP-HPLC determination of the lipophilicity of bispyridinium reactivators of acetylcholinesterase bearing a but-2-ene connecting linker

Kamil Musilek, Josef Jampilek, Jiri Dohnal, Daniel Jun, Frank Gunn-Moore, Martin Dolezal, Kamil Kuca

Journal:

Analytical and Bioanalytical Chemistry

Année:

2008

Langue:

english

Fichier:

PDF, 142 KB

english, 2008

29

Fluctuation in the ergosterol and deoxynivalenol content in barley and malt during malting process

Vlastimil Dohnal, Alena Jezkova, Lucie Pavlikova, Kamil Musilek, Daniel Jun, Kamil Kuca

Journal:

Analytical and Bioanalytical Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 183 KB

english, 2010

30

Selected AChE reactivators in different crystalline environment: salts and enzyme

Agnieszka Skórska-Stania, Magdalena Śliwa, Kamil Musilek, Kamil Kuca, Josef Jampilek, Robert Musiol, Barbara J. Oleksyn, Jiri Dohnal

Journal:

Structural Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 513 KB

english, 2010

31

Methylacridinium and its Cholinergic Properties

Ondrej Soukup, Jan Proska, Jiri Binder, Jana Zdarova Karasova, Gunnar Tobin, Daniel Jun, Jan Marek, Kamil Musílek, Josef Fusek, Kamil Kuca

Journal:

Neurotoxicity Research

Année:

2009

Langue:

english

Fichier:

PDF, 288 KB

english, 2009

32

Synthesis of the novel series of bispyridinium compounds bearing (E)-but-2-ene linker and evaluation of their reactivation activity against chlorpyrifos-inhibited acetylcholinesterase

Kamil Musilek, Kamil Kuca, Daniel Jun, Vlastimil Dohnal, Martin Dolezal

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2006

Langue:

english

Fichier:

PDF, 147 KB

english, 2006

33

Synthesis of asymmetrical bispyridinium compounds bearing cyano-moiety and evaluation of their reactivation activity against tabun and paraoxon-inhibited acetylcholinesterase

Kamil Musilek, Ondrej Holas, Kamil Kuca, Daniel Jun, Vlastimil Dohnal, Martin Dolezal

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2006

Langue:

english

Fichier:

PDF, 141 KB

english, 2006

34

Evaluation of the Neuroprotective Efficacy of Newly Developed Oximes (K206, K269) and Currently Available Oximes (Obidoxime, HI-6) in Cyclosarin-Poisoned Rats

Jiri Kassa, Jana Zdarova Karasova, Jiri Bajgar, Sandra Tesarova, Kamil Kuca, Kamil Musilek

Journal:

Basic & Clinical Pharmacology & Toxicology

Année:

2009

Langue:

english

Fichier:

PDF, 103 KB

english, 2009

35

Reactivation of Human Brain Homogenate Cholinesterases Inhibited by Tabun using Newly Developed Oximes K117 and K127

Kamil Kuca, Jiri Cabal, Yung Sik Jung, Kamil Musilek, Ondrej Soukup, Daniel Jun, Miroslav Pohanka, Lucie Musilova, Jana Karasová, Ladislav Novotný, Martina Hrabinova

Journal:

Basic & Clinical Pharmacology & Toxicology

Année:

2009

Langue:

english

Fichier:

PDF, 135 KB

english, 2009

36

A Comparison of Neuroprotective Efficacy of the Oxime K203 and its Fluorinated Analogue (KR-22836) with Obidoxime in Tabun-Poisoned Rats

Jiri Kassa, Jana Zdarova Karasova, Sandra Tesarova, Kamil Musilek, Kamil Kuca, Young-Sik Jung

Journal:

Basic & Clinical Pharmacology & Toxicology

Année:

2010

Langue:

english

Fichier:

PDF, 122 KB

english, 2010

37

Reactivation kinetics of a homologous series of bispyridinium bis-oximes with nerve agent-inhibited human acetylcholinesterase

Franz Worek, Jens von der Wellen, Kamil Musilek, Kamil Kuca, Horst Thiermann

Journal:

Archives of Toxicology

Année:

2012

Langue:

english

Fichier:

PDF, 649 KB

english, 2012

38

Synthesis and in vitro evaluation of 7-methoxy-N-(pent-4-enyl)-1,2,3,4-tetrahydroacridin-9-amine—new tacrine derivate with cholinergic properties

Jan Korabecny, Kamil Musilek, Filip Zemek, Anna Horova, Ondrej Holas, Eugenie Nepovimova, Veronika Opletalova, Jana Hroudova, Zdenek Fisar, Young-Sik Jung, Kamil Kuca

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 535 KB

english, 2011

39

A Comparison of the Efficacy of Newly Developed Reversible Inhibitors of Acetylcholinesterase with Commonly Used Pyridostigmine as Pharmacological Pre-Treatment of Soman-Poisoned Mice

Jiri Kassa, Kamil Musilek, Marketa Koomlova, Jiri Bajgar

Journal:

Basic & Clinical Pharmacology & Toxicology

Année:

2012

Langue:

english

Fichier:

PDF, 152 KB

english, 2012

40

The progress in the cholinesterase quantification methods

Holas, Ondrej, Musilek, Kamil, Pohanka, Miroslav, Kuca, Kamil

Journal:

Expert Opinion on Drug Discovery

Année:

2012

Langue:

english

Fichier:

PDF, 644 KB

english, 2012

41

Reactivation of VX-inhibited AChE by novel oximes having two oxygen atoms in the linker

Kamil Kuca, Jiri Cabal, Daniel Jun, Kamil Musilek, Ondrej Soukup, Miroslav Pohanka, Jaroslav Pejchal, Kyung-Ae Oh, Garp Yeol Yang, Young-Sik Jung

Journal:

Environmental Toxicology and Pharmacology

Année:

2010

Langue:

english

Fichier:

PDF, 211 KB

english, 2010

42

Passive diffusion of acetylcholinesterase oxime reactivators through the blood–brain barrier: Influence of molecular structure

Jana Zdarova Karasova, Miroslav Pohanka, Kamil Musilek, Filip Zemek, Kamil Kuca

Journal:

Toxicology in Vitro

Année:

2010

Langue:

english

Fichier:

PDF, 2.47 MB

english, 2010

43

In vitro effects of acetylcholinesterase reactivators on monoamine oxidase activity

Zdeněk Fišar, Jana Hroudová, Jan Korábečný, Kamil Musílek, Kamil Kuča

Journal:

Toxicology Letters

Année:

2011

Langue:

english

Fichier:

PDF, 194 KB

english, 2011

44

Time-Dependent Changes of Oxime K027 Concentrations in Different Parts of Rat Central Nervous System

Jana Zdarova Karasova, Filip Zemek, Kamil Musilek, Kamil Kuca

Journal:

Neurotoxicity Research

Année:

2013

Langue:

english

Fichier:

PDF, 251 KB

english, 2013

45

Structure-activity relationship for the reactivators of acetylcholinesterase inhibited by nerve agent VX

Kamil Kuca, Daniel Jun, Kamil Musilek, Jiri Bajgar

Journal:

Toxicology Letters

Année:

2006

Langue:

english

Fichier:

PDF, 77 KB

english, 2006

46

Reactivators of acetylcholinesterase for organophosphorus pesticide intoxication—May we replace pralidoxime?

Kamil Musilek, Ondrej Holas, Veronika Opletalova, Daniel Jun, Kamil Kuca

Journal:

Toxicology Letters

Année:

2008

Langue:

english

Fichier:

PDF, 85 KB

english, 2008

47

Newly developed oximes K117 and K127—Reactivation of human brain cholinesterases inhibited by tabun

Jan Marek, Kamil Kuca, Jiri Cabal, Kamil Musilek, Jana Karasova, Y.S. Jung, Daniel Jun, Miroslav Pohanka

Journal:

Toxicology Letters

Année:

2009

Langue:

english

Fichier:

PDF, 75 KB

english, 2009

48

Small quaternary AChE inhibitors—Implication for pretreatment of OP poisoning or MG treatment

Kamil Musilek, Marketa Komloova, Ondrej Holas, Miroslav Pohanka, Veronika Opletalova, Martin Dolezal, Kamil Kuca

Journal:

Toxicology Letters

Année:

2009

Langue:

english

Fichier:

PDF, 83 KB

english, 2009

49

Effect of 10 oxime cholinesterase reactivators on cyclosarin-intoxicated rats

Jana Zdarova Karasova, Jiri Kassa, Kamil Musilek, Miroslav Pohanka, Kamil Kuca

Journal:

Toxicology Letters

Année:

2009

Langue:

english

Fichier:

PDF, 94 KB

english, 2009

50

Preparation of the Pyridinium Salts Differing in the Length of the N-Alkyl Substituent

Marek, Jan, Stodulka, Petr, Cabal, Jiri, Soukup, Ondrej, Pohanka, Miroslav, Korabecny, Jan, Musilek, Kamil, Kuca, Kamil

Journal:

Année:

2010

Langue:

english

Fichier:

PDF, 99 KB

english, 2010